Heat shock protein 90: inhibitors in clinical trials

J Med Chem. 2010 Jan 14;53(1):3-17. doi: 10.1021/jm9004708.
No abstract available

MeSH terms

  • Animals
  • Benzamides / chemical synthesis
  • Benzamides / chemistry
  • Benzamides / pharmacology*
  • Benzoquinones / chemical synthesis
  • Benzoquinones / chemistry
  • Benzoquinones / pharmacology*
  • Clinical Trials as Topic*
  • Drug Design
  • Drug Screening Assays, Antitumor
  • HSP90 Heat-Shock Proteins / antagonists & inhibitors*
  • HSP90 Heat-Shock Proteins / metabolism
  • Humans
  • Lactams, Macrocyclic / chemical synthesis
  • Lactams, Macrocyclic / chemistry
  • Lactams, Macrocyclic / pharmacology*
  • Molecular Structure
  • Purines / chemical synthesis
  • Purines / chemistry
  • Purines / pharmacology*
  • Resorcinols / chemical synthesis
  • Resorcinols / chemistry
  • Resorcinols / pharmacology*
  • Structure-Activity Relationship

Substances

  • Benzamides
  • Benzoquinones
  • HSP90 Heat-Shock Proteins
  • Lactams, Macrocyclic
  • Purines
  • Resorcinols
  • 17-(dimethylaminoethylamino)-17-demethoxygeldanamycin
  • tanespimycin
  • benzamide
  • purine
  • resorcinol